| Bioengineered PLGA-chitosan nanoparticles for brain targeted intranasal delivery of antiepileptic TRH analogues NW S. Kaur, P. Manhas, A. Swami, R. Bhandari, K.K. Sharma, R. Jain, R. Kumar ... Chemical Engineering Journal 346, 630, 2018 | 67 | 2018 |
| Peptide-based drug discovery: current status and recent advances K Sharma, KK Sharma, A Sharma, R Jain Drug Discovery Today 28 (2), 103464, 2023 | 46 | 2023 |
| Room Temperature N-Arylation of Amino Acids and Peptides Using Copper (I) and β-diketone KK Sharma, S Sharma, A Kudwal, R Jain Organic & Biomolecular Chemistry 13, 4637-4641, 2015 | 46 | 2015 |
| Metal-free synthesis of N-fused heterocyclic iodides via C–H functionalization mediated by tert-butylhydroperoxide KK Sharma, DI Patel, R Jain Chemical Communications 51 (82), 15129-15132, 2015 | 44 | 2015 |
| Rapid microwave-assisted solution-phase peptide synthesis A Mahindra, KK Sharma, R Jain Tetrahedron Letters 53 (51), 6931-6935, 2012 | 40 | 2012 |
| Discovery of a Membrane-Active, Ring-Modified Histidine Containing Ultrashort Amphiphilic Peptide That Exhibits Potent Inhibition of Cryptococcus neoformans KK Sharma, IK Maurya, SI Khan, MR Jacob, V Kumar, K Tikoo, R Jain Journal of Medicinal Chemistry 60 (15), 6607-6621, 2017 | 36 | 2017 |
| Tyr1-ψ[(Z)CF=CH]-Gly2 Fluorinated Peptidomimetic Improves Distribution and Metabolism Properties of Leu-Enkephalin RA Altman, KK Sharma, LG Rajewski, PC Toren, MJ Baltezor, M Pal, ... ACS Chemical Neuroscience 9 (7), 1735, 2018 | 35 | 2018 |
| Microwave-assisted solution phase peptide synthesis in neat water A Mahindra, K Nooney, S Uraon, KK Sharma, R Jain RSC Advances 3 (37), 16810-16816, 2013 | 28 | 2013 |
| Regioselective copper-catalyzed N(1)-(hetero)arylation of protected histidine Krishna K Sharma, Meenakshi Mandloi, Rahul Jain Organic and Biomolecular Chemistry 14, 8937-8941, 2016 | 24 | 2016 |
| Synthesis and antimicrobial activities of His (2-aryl)-Arg and Trp-His (2-aryl) classes of dipeptidomimetics A Mahindra, KK Sharma, D Rathore, SI Khan, MR Jacob, R Jain MedChemComm 5 (5), 671-676, 2014 | 24 | 2014 |
| Modified Histidine Containing Amphipathic Ultrashort Antifungal Peptide, His[2-p-(n-butyl)phenyl]-Trp-Arg-OMe Exhibits Potent Anticryptococcal Activity KK Sharma, R Ravi, IK Maurya, A Kapadia, SI Khan, V Kumar, K Tikoo, ... European Journal of Medicinal Chemistry 223 (2021), 113635, 2021 | 22 | 2021 |
| Copper-catalyzed N-(hetero)arylation of amino acids in water KK Sharma, M Mandloi, N Rai, R Jain RSC Advances 6 (99), 96762-96767, 2016 | 21 | 2016 |
| Synthesis, stability and mechanistic studies of potent anticryptococcal hexapeptides K Shenmar, KK Sharma, N Wangoo, IK Maurya, V Kumar, SI Khan, ... European Journal of Medicinal Chemistry 132, 192, 2017 | 14 | 2017 |
| New Structural Classes of Antimalarials GK Rathod, M Jain, KK Sharma, S Das, A Basak, R Jain European Journal of Medicinal Chemistry 242, 114653, 2022 | 13 | 2022 |
| Regioselective Access to 1,2-Diarylhistidines through the Copper-Catalyzed N1-Arylation of 2-Arylhistidines KK Sharma, M Mandloi, R Jain European Journal of Organic Chemistry 2017 (5), 984–988, 2017 | 13 | 2017 |
| The Meta-Position of Phe4 in Leu-Enkephalin Regulates Potency, Selectivity, Functional Activity, and Signaling Bias at the Delta and Mu Opioid Receptors RJ Cassell, KK Sharma, H Su, BR Cummins, H Cui, KL Mores, AT Blaine, ... Molecules 24, 4542, 2019 | 11 | 2019 |
| Synthetic Amino Acids-Derived Peptides Targets Cryptococcus neoformans by Inducing Cell Membrane Disruption K Sharma, S Aaghaz, I Maurya, KK Sharma, SM Rudramurth, S Singh, ... Bioorganic Chemistry 130 (2023), 106252, 2023 | 10 | 2023 |
| Effect of C-terminus amidation of Aβ39-42 fragment derived peptides as potential inhibitors of Aβ aggregation A Kapadia, A Patel, KK Sharma, IK Maurya, V Singh, M Khullar, R Jain RSC Advances 10 (25), 27137-27151, 2020 | 10 | 2020 |
| A General Strategy to Install Amidine Functional Groups Along the Peptide Backbone EA O’Brien, KK Sharma, J Byerly-Duke, LA Camacho III, B VanVeller Journal of the American Chemical Society 144 (49), 22397−22402, 2022 | 9 | 2022 |
| Thyrotropin-Releasing Hormone Loaded and Chitosan Engineered Polymeric Nanoparticles: Towards Effective Delivery of Neuropeptides S Kaur, A Bhararia, KK Sharma, S Mittal, R Jain, N Wangoo, RK Sharma Journal of Nanoscience and Nanotechnology 16 (5), 5324-5332, 2016 | 9 | 2016 |
Rahul JainProfessor of Medicinal Chemistry, National Institute of Pharmaceutical Education and ResearchDirección de correo verificada de niper.ac.in
