| Insights into the mechanism of partial agonism: crystal structures of the peroxisome proliferator-activated receptor γ ligand-binding domain in the complex with two … G Pochetti, C Godio, N Mitro, D Caruso, A Galmozzi, S Scurati, F Loiodice, ... Journal of Biological Chemistry 282 (23), 17314-17324, 2007 | 140 | 2007 |
| Crystal structure of the peroxisome proliferator-activated receptor γ (PPARγ) ligand binding domain complexed with a novel partial agonist: a new region of the hydrophobic … R Montanari, F Saccoccia, E Scotti, M Crestani, C Godio, F Gilardi, ... Journal of medicinal chemistry 51 (24), 7768-7776, 2008 | 126 | 2008 |
| Resveratrol and its metabolites bind to PPARs E Calleri, G Pochetti, KSS Dossou, A Laghezza, R Montanari, D Capelli, ... ChemBioChem 15 (8), 1154-1160, 2014 | 95 | 2014 |
| Extra Binding Region Induced by Non-Zinc Chelating Inhibitors into the S1′ Subsite of Matrix Metalloproteinase 8 (MMP-8) G Pochetti, R Montanari, C Gege, C Chevrier, AG Taveras, F Mazza Journal of medicinal chemistry 52 (4), 1040-1049, 2009 | 91 | 2009 |
| Structural insight into the stereoselective inhibition of MMP-8 by enantiomeric sulfonamide phosphonates G Pochetti, E Gavuzzo, C Campestre, M Agamennone, P Tortorella, ... Journal of medicinal chemistry 49 (3), 923-931, 2006 | 87 | 2006 |
| Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode D Capelli, C Cerchia, R Montanari, F Loiodice, P Tortorella, A Laghezza, ... Scientific reports 6 (1), 34792, 2016 | 82 | 2016 |
| Betulinic acid is a PPARγ antagonist that improves glucose uptake, promotes osteogenesis and inhibits adipogenesis G Brusotti, R Montanari, D Capelli, G Cattaneo, A Laghezza, P Tortorella, ... Scientific reports 7 (1), 5777, 2017 | 77 | 2017 |
| γ-Turn conformation induced by α, α-disubstituted amino acids with a cyclic six-membered side chain MP Paradisi, I Torrini, GP Zecchini, G Lucente, E Gavuzzo, F Mazza, ... Tetrahedron 51 (8), 2379-2386, 1995 | 71 | 1995 |
| N-Hydroxyurea as zinc binding group in matrix metalloproteinase inhibition: mode of binding in a complex with MMP-8 C Campestre, M Agamennone, P Tortorella, S Preziuso, A Biasone, ... Bioorganic & medicinal chemistry letters 16 (1), 20-24, 2006 | 62 | 2006 |
| Synthesis and properties of chemotactic peptide analogs: II. HCO‐Met‐Leu‐Phe‐OMe analogs containing cyclic α, α‐disubstituted amino acids as Met and Phe mimicking residues I Torrini, GP Zecchini, MP Paradisi, G Lucente, E Gavuzzo, F Mazza, ... International Journal of Peptide and Protein Research 38 (6), 495-504, 1991 | 61 | 1991 |
| Two crystal structures of human neutrophil collagenase, one complexed with a primed-and the other with an unprimed-side inhibitor: implications for drug design E Gavuzzo, G Pochetti, F Mazza, C Gallina, B Gorini, S D'Alessio, ... Journal of medicinal chemistry 43 (18), 3377-3385, 2000 | 58 | 2000 |
| Crystal phases obtained from aqueous solutions of sodium dodecyl sulfate. The structure of a monoclinic phase of sodium dodecyl sulfate hemihydrate VM Coiro, F Mazza, G Pochetti Acta Crystallographica Section C: Crystal Structure Communications 42 (8 …, 1986 | 58 | 1986 |
| Structure of a triclinic phase of sodium dodecyl sulfate monohydrate. A comparison with other sodium dodecyl sulfate crystal phases VM Coiro, M Manigrasso, F Mazza, G Pochetti Acta Crystallographica Section C: Crystal Structure Communications 43 (5 …, 1987 | 56 | 1987 |
| Synthesis, characterization and biological evaluation of ureidofibrate-like derivatives endowed with peroxisome proliferator-activated receptor activity L Porcelli, F Gilardi, A Laghezza, L Piemontese, N Mitro, A Azzariti, ... Journal of medicinal chemistry 55 (1), 37-54, 2012 | 55 | 2012 |
| Structural insight into peroxisome proliferator-activated receptor γ binding of two ureidofibrate-like enantiomers by molecular dynamics, cofactor interaction analysis, and … G Pochetti, N Mitro, A Lavecchia, F Gilardi, N Besker, E Scotti, M Aschi, ... Journal of medicinal chemistry 53 (11), 4354-4366, 2010 | 55 | 2010 |
| 2 Å X-ray structure of adamalysin II complexed with a peptide phosphonate inhibitor adopting a retro-binding mode M Cirilli, C Gallina, E Gavuzzo, C Giordano, FX Gomis-Rüth, B Gorini, ... FEBS letters 418 (3), 319-322, 1997 | 49 | 1997 |
| New 2-aryloxy-3-phenyl-propanoic acids as peroxisome proliferator-activated receptors α/γ dual agonists with improved potency and reduced adverse effects on skeletal muscle … G Fracchiolla, A Laghezza, L Piemontese, P Tortorella, F Mazza, ... Journal of medicinal chemistry 52 (20), 6382-6393, 2009 | 46 | 2009 |
| Crystal structure, conformation, and potential energy calculations the chemotactic peptide N‐ formyl‐l‐Met‐l‐Leu‐l‐Phe‐OMe E GAVUZZO, F MAZZA, G POCHETTI, A SCATTURIN International Journal of Peptide and Protein Research 34 (5), 409-415, 1989 | 46 | 1989 |
| LT175 is a novel PPARα/γ ligand with potent insulin-sensitizing effects and reduced adipogenic properties F Gilardi, M Giudici, N Mitro, O Maschi, U Guerrini, G Rando, A Maggi, ... Journal of Biological Chemistry 289 (10), 6908-6920, 2014 | 45 | 2014 |
| Structure and conformation of peptides containing the sulphonamide junction: I. N‐acetyl‐tauryl‐l‐phenylalanine methyl ester A Calcagni, E Gavuzzo, G Lucente, F Mazza, G Pochetti, D Rossi International Journal of Peptide and Protein Research 34 (4), 319-324, 1989 | 45* | 1989 |
