Synthesis and SAR Studies of 1H-Pyrrolo[2,3-b]pyridine-2-carboxamides as Phosphodiesterase 4B (PDE4B) Inhibitors AK Vadukoot, S Sharma, CD Aretz, S Kumar, N Gautam, Y Alnouti, ... ACS Medicinal Chemistry Letters 11 (10), 1848-1854, 2020 | 15 | 2020 |
Discovery of Small Molecule Renal Outer Medullary Potassium (ROMK) Channel Inhibitors: A Brief History of Medicinal Chemistry Approaches To Develop Novel Diuretic Therapeutics … CD Aretz, AK Vadukoot, CR Hopkins Journal of Medicinal Chemistry 62 (19), 8682-8694, 2019 | 7 | 2019 |
Cyclopentane Formation from Flexible Precursors Using Samarium (II) Reagents CD Aretz, H Escobedo, BJ Cowen European Journal of Organic Chemistry 2018 (16), 1880-1884, 2018 | 7 | 2018 |
Further SAR on the (Phenylsulfonyl)piperazine Scaffold as Inhibitors of the Aedes aegypti Kir1 (AeKir) Channel and Larvicides CD Aretz, SV Kharade, K Chronister, R Rusconi Trigueros, ... ChemMedChem 16 (2), 319-327, 2021 | 5 | 2021 |
Discovery and Characterization of 2-Nitro-5-(4-(phenylsulfonyl)piperazin-1-yl)-N-(pyridin-4-ylmethyl)anilines as Novel Inhibitors of the Aedes aegypti Kir1 (AeKir1 … CD Aretz, MJ Morwitzer, AG Sanford, AM Hogan, MV Portillo, SV Kharade, ... ACS infectious diseases 5 (6), 917-931, 2019 | 5 | 2019 |
Mechanism of SmI2 Reduction of 5-Bromo-6-oxo-6-phenylhexyl Methanesulfonate Studied by Spin Trapping with 2-Methyl-2-nitrosopropane CD Aretz, JE McPeak, GR Eaton, SS Eaton, BJ Cowen The Journal of Organic Chemistry 83 (17), 10688-10692, 2018 | 5 | 2018 |
Synthesis and biological characterization of a series of 2-sulfonamidebenzamides as allosteric modulators of mrgX1 S Sharma, Q Peng, AK Vadukoot, CD Aretz, AA Jensen, AI Wallick, ... ACS Medicinal Chemistry Letters 13 (5), 841-847, 2022 | 1 | 2022 |
Further synthesis and biological characterization of a series of 2-sulfonamidebenzamides as allosteric modulators of MrgX1 S Sharma, Q Peng, A Vadukoot, C Aretz, A Jensen, A Wallick, X Dong, ... | | 2021 |
Discovery, synthesis and biological characterization of a series of N-(1-(1, 1-dioxidotetrahydrothiophen-3-yl)-3-methyl-1 H-pyrazol-5-yl) acetamide ethers as novel GIRK1/2 … S Sharma, L Lesiak, CD Aretz, Y Du, S Kumar, N Gautam, Y Alnouti, ... RSC Medicinal Chemistry 12 (8), 1366-1373, 2021 | | 2021 |
Discovery and characterization of a novel class of phenylsulfonylpiperazine containing compounds as inhibitors of the Aedes aegypti Kir1 (AeKir1) potassium … JB Mccarthey, CD Aretz, MD Morwitzer, AG Sanford, AM Hogan, ... The FASEB Journal 33 (S1), 862.8-862.8, 2019 | | 2019 |
Selective Carbon-Carbon Bond Formation Promoted by Divalent Samarium Reagents CDJ Aretz | | 2018 |
Stereoselective samarium diiodide promoted carbon carbon bond forming reactions C Aretz, H Escobedo, B Cowen ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 249, 2015 | | 2015 |