Solid-phase synthesis of isocoumarins: a traceless halocyclization approach M Peuchmaur, V Lisowski, C Gandreuil, LT Maillard, J Martinez, ... The Journal of Organic Chemistry 74 (11), 4158-4165, 2009 | 69 | 2009 |
Helical oligomers of Thiazole‐based γ‐amino acids: synthesis and structural studies L Mathieu, B Legrand, C Deng, L Vezenkov, E Wenger, C Didierjean, ... Angewandte Chemie International Edition 52 (23), 6006-6010, 2013 | 65 | 2013 |
1, 2, 4‐Triazole‐3‐thione Compounds as Inhibitors of Dizinc Metallo‐β‐lactamases L Sevaille, L Gavara, C Bebrone, F De Luca, L Nauton, M Achard, ... ChemMedChem 12 (12), 972-985, 2017 | 59 | 2017 |
Synthesis and anti-Candida activity of novel 2-hydrazino-1,3-thiazole derivatives LT Maillard, S Bertout, O Quinonéro, G Akalin, G Turan-Zitouni, ... Bioorganic & medicinal chemistry letters 23 (6), 1803-1807, 2013 | 52 | 2013 |
Imidazopyridine-fused [1, 3]-diazepinones: synthesis and antiproliferative activity A Gallud, O Vaillant, LT Maillard, DP Arama, J Dubois, M Maynadier, ... European Journal of Medicinal Chemistry 75, 382-390, 2014 | 49 | 2014 |
Thiazole‐Based γ‐Building Blocks as Reverse‐Turn Mimetic to Design a Gramicidin S Analogue: Conformational and Biological Evaluation B Legrand, L Mathieu, A Lebrun, S Andriamanarivo, V Lisowski, ... Chemistry–A European Journal 20 (22), 6713-6720, 2014 | 44 | 2014 |
Selective C-Acylation of 2-Aminoimidazo[1,2-a]pyridine: Application to the Synthesis of Imidazopyridine-Fused [1,3]Diazepinones N Masurier, R Aruta, V Gaumet, S Denoyelle, E Moreau, V Lisowski, ... The Journal of Organic Chemistry 77 (7), 3679-3685, 2012 | 32 | 2012 |
A New Supported Reagent for the Parallel Synthesis of Primary and Secondary O-Alkyl Hydroxylamines through a Base-Catalyzed Mitsunobu Reaction LT Maillard, M Benohoud, P Durand, B Badet The Journal of Organic Chemistry 70 (16), 6303-6312, 2005 | 32 | 2005 |
Pyrido-imidazodiazepinones as a new class of reversible inhibitors of human kallikrein 7 DP Arama, F Soualmia, V Lisowski, JF Longevial, E Bosc, LT Maillard, ... European journal of medicinal chemistry 93, 202-213, 2015 | 25 | 2015 |
A tandem aza-Friedel–Crafts reaction/Hantzsch cyclization: a simple procedure to access polysubstituted 2-amino-1, 3-thiazoles G Chaubet, LT Maillard, J Martinez, N Masurier Tetrahedron 67 (26), 4897-4904, 2011 | 24 | 2011 |
Helical γ‐peptide foldamers as dual inhibitors of amyloid‐β Peptide and islet amyloid polypeptide oligomerization and fibrillization J Kaffy, C Berardet, L Mathieu, B Legrand, M Taverna, F Halgand, ... Chemistry–A European Journal 26 (64), 14612-14622, 2020 | 23 | 2020 |
Catalytic foldamers: When the structure guides the function B Legrand, J Aguesseau-Kondrotas, M Simon, L Maillard Catalysts 10 (6), 700, 2020 | 23 | 2020 |
How to deal with weak interactions in noncovalent complexes analyzed by electrospray mass spectrometry: cyclopeptidic inhibitors of the nuclear receptor coactivator 1-STAT6 D Touboul, L Maillard, A Grässlin, R Moumne, M Seitz, J Robinson, ... Journal of the American Society for Mass Spectrometry 20, 303-311, 2009 | 19 | 2009 |
Prospect of Thiazole‐based γ‐Peptide Foldamers in Enamine Catalysis: Exploration of the Nitro‐Michael Addition J Aguesseau‐Kondrotas, M Simon, B Legrand, JL Bantigniès, YK Kang, ... Chemistry–A European Journal 25 (30), 7396-7401, 2019 | 18 | 2019 |
Imidazopyridine-fused [1, 3]-diazepinones part 2: structure-activity relationships and antiproliferative activity against melanoma cells V Bellet, L Lichon, DP Arama, A Gallud, V Lisowski, LT Maillard, M Garcia, ... European Journal of Medicinal Chemistry 125, 1225-1234, 2017 | 17 | 2017 |
FT-IR and NMR structural markers for thiazole-based γ-peptide foldamers C Bonnel, B Legrand, JL Bantignies, H Petitjean, J Martinez, N Masurier, ... Organic & Biomolecular Chemistry 14 (37), 8664-8669, 2016 | 17 | 2016 |
Monitoring enzyme‐catalyzed production of glucosamine‐6P by matrix‐assisted laser desorption/ionization time‐of‐flight mass spectrometry: a new enzymatic assay for glucosamine … LT Maillard, V Guérineau, MA Badet‐Denisot, B Badet, O Laprévote, ... Rapid Communications in Mass Spectrometry: An International Journal Devoted …, 2006 | 16 | 2006 |
Tailoring the physicochemical properties of antimicrobial peptides onto a thiazole-based γ-peptide foldamer C Bonnel, B Legrand, M Simon, M Clavié, A Masnou, E Jumas-Bilak, ... Journal of Medicinal Chemistry 63 (17), 9168-9180, 2020 | 15 | 2020 |
Molecular Characterization of the NCoA‐1–STAT 6 Interaction M Seitz, LT Maillard, D Obrecht, JA Robinson ChemBioChem 9 (8), 1318-1322, 2008 | 14 | 2008 |
Can Heterocyclic γ‐Peptides Provide Polyfunctional Platforms for Synthetic Glycocluster Construction? M Simon, LMA Ali, K El Cheikh, J Aguesseau, M Gary‐Bobo, M Garcia, ... Chemistry–A European Journal 24 (44), 11426-11432, 2018 | 12 | 2018 |