| Cell-permeable nanobodies for targeted immunolabelling and antigen manipulation in living cells HD Herce, D Schumacher, AFL Schneider, AK Ludwig, FA Mann, M Fillies, ... Nature chemistry 9 (8), 762-771, 2017 | 257 | 2017 |
| Cysteine‐Selective Phosphonamidate Electrophiles for Modular Protein Bioconjugations MA Kasper, M Glanz, A Stengl, M Penkert, S Klenk, T Sauer, ... Angewandte Chemie International Edition 58 (34), 11625-11630, 2019 | 101 | 2019 |
| LNA-enhanced DNA FIT-probes for multicolour RNA imaging F Hövelmann, I Gaspar, J Chamiolo, M Kasper, J Steffen, A Ephrussi, ... Chemical Science 7 (1), 128-135, 2016 | 82 | 2016 |
| Ethynylphosphonamidates for the Rapid and Cysteine‐Selective Generation of Efficacious Antibody–Drug Conjugates MA Kasper, A Stengl, P Ochtrop, M Gerlach, T Stoschek, D Schumacher, ... Angewandte Chemie International Edition 58 (34), 11631-11636, 2019 | 59 | 2019 |
| Vinylphosphonites for Staudinger-induced chemoselective peptide cyclization and functionalization MA Kasper, M Glanz, A Oder, P Schmieder, JP von Kries, ... Chemical Science 10 (25), 6322-6329, 2019 | 57 | 2019 |
| Protein modification of lysine with 2-(2-styrylcyclopropyl) ethanal C Apel, MA Kasper, CE Stieger, CPR Hackenberger, M Christmann Organic letters 21 (24), 10043-10047, 2019 | 21 | 2019 |
| β‐Carotene Revisited by Transient Absorption and Stimulated Raman Spectroscopy M Quick, MA Kasper, C Richter, R Mahrwald, AL Dobryakov, ... ChemPhysChem 16 (18), 3824-3835, 2015 | 20 | 2015 |
| Bis (arylmethyl)-substituted unsymmetrical phosphites for the synthesis of lipidated peptides via Staudinger-phosphite reactions N Nischan, MA Kasper, T Mathew, CPR Hackenberger Organic & Biomolecular Chemistry 14 (31), 7500-7508, 2016 | 18 | 2016 |
| N‐Hydroxysuccinimide‐Modified Ethynylphosphonamidates Enable the Synthesis of Configurationally Defined Protein Conjugates MA Kasper, M Gerlach, AFL Schneider, C Groneberg, P Ochtrop, S Boldt, ... ChemBioChem 21 (1-2), 113-119, 2020 | 15 | 2020 |
| Cysteinselektive phosphonamidatbasierte Elektrophile für modulare Biokonjugationen MA Kasper, M Glanz, A Stengl, M Penkert, S Klenk, T Sauer, ... Angewandte Chemie 131 (34), 11751-11756, 2019 | 15 | 2019 |
| TuPPL: Tub-tag mediated C-terminal protein–protein-ligation using complementary click-chemistry handles A Stengl, M Gerlach, MA Kasper, CPR Hackenberger, H Leonhardt, ... Organic & Biomolecular Chemistry 17 (20), 4964-4969, 2019 | 12 | 2019 |
| The mechanism behind enhanced reactivity of unsaturated phosphorus (v) electrophiles towards thiols Y Park, AL Baumann, H Moon, S Byrne, MA Kasper, S Hwang, H Sun, ... Chemical Science 12 (23), 8141-8148, 2021 | 10 | 2021 |
| Targeting FLT3 with a new-generation antibody-drug conjugate in combination with kinase inhibitors for treatment of AML M Roas, B Vick, MA Kasper, M Able, H Polzer, M Gerlach, E Kremmer, ... Blood, The Journal of the American Society of Hematology 141 (9), 1023-1035, 2023 | 8 | 2023 |
| Compact hydrophilic electrophiles enable highly efficacious high DAR ADCs with excellent in vivo PK profile P Ochtrop, J Jahzerah, P Machui, I Mai, D Schumacher, J Helma, ... Chemical Science 14 (9), 2259-2266, 2023 | 5 | 2023 |
| Bis‐ethynylphosphonamidates as an Modular Conjugation Platform to Generate Multi‐Functional Protein‐and Antibody‐Drug‐Conjugates MA Kasper, L Lassak, AM Vogl, I Mai, J Helma, D Schumacher, ... European Journal of Organic Chemistry 2022 (10), e202101389, 2022 | 5 | 2022 |
| (3+ 2)‐Cyclization Reactions of Unsaturated Phosphonites with Aldehydes and Thioketones DS Munasinghe, MA Kasper, R Jasiński, K Kula, M Palusiak, M Celeda, ... Chemistry–A European Journal 29 (33), e202300806, 2023 | 2 | 2023 |
| Tub-010, a novel antibody-drug-conjugate with reduced nonspecific toxicity profile based on tub-tag technology widens the therapeutic window for the treatment of CD30+ Malignancies M Gerlach, S Schmitt, P Cyprys, MA Kasper, I Mai, MH Vermeer, ... Blood 140 (Supplement 1), 9397-9398, 2022 | 1 | 2022 |
| Chemoselective thiol-conjugation with alkene or alkyne-phosphonamidates C Hackenberger, MA Kasper, M Glanz, T Sauer, D Schumacher, ... US Patent 11,161,873, 2021 | 1 | 2021 |
| Chemoselective synthesis of functional drug conjugates MA Kasper Humboldt-Universität zu Berlin, 2020 | 1 | 2020 |
| TUB-040, a novel Napi2b-targeting ADC built with ethynylphosphonamidate conjugation chemistry, demonstrates high and long-lasting anti-tumor efficacy via Topoisomerase-I … S Schmitt, I Mai, P Machui, S Herterich, D Hauswald, P Ochtrop, P Cyprys, ... Cancer Research 84 (6_Supplement), 2622-2622, 2024 | | 2024 |
