| Expanding Pd-catalyzed C− N bond-forming processes: the first amidation of aryl sulfonates, aqueous amination, and complementarity with Cu-catalyzed reactions X Huang, KW Anderson, D Zim, L Jiang, A Klapars, SL Buchwald Journal of the American Chemical Society 125 (22), 6653-6655, 2003 | 929 | 2003 |
| The selective reaction of aryl halides with KOH: synthesis of phenols, aromatic ethers, and benzofurans KW Anderson, T Ikawa, RE Tundel, SL Buchwald Journal of the American Chemical Society 128 (33), 10694-10695, 2006 | 552 | 2006 |
| General catalysts for the Suzuki–Miyaura and Sonogashira coupling reactions of aryl chlorides and for the coupling of challenging substrate combinations in water KW Anderson, SL Buchwald Angewandte Chemie 117 (38), 6329-6333, 2005 | 495 | 2005 |
| A highly active catalyst for Suzuki-Miyaura cross-coupling reactions of heteroaryl compounds KL Billingsley, KW Anderson, SL Buchwald ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH- 45 (21), 3484, 2006 | 417 | 2006 |
| Monodentate Phosphines Provide Highly Active Catalysts for Pd‐Catalyzed C N Bond‐Forming Reactions of Heteroaromatic Halides/Amines and (H) N‐Heterocycles KW Anderson, RE Tundel, T Ikawa, RA Altman, SL Buchwald Angewandte Chemie International Edition 45 (39), 6523-6527, 2006 | 375 | 2006 |
| Sequential Cu-Catalyzed Amidation-Base-Mediated Camps Cyclization: A Two-Step Synthesis of 2-Aryl-4-quinolones from o-Halophenones CP Jones, KW Anderson, SL Buchwald The Journal of organic chemistry 72 (21), 7968-7973, 2007 | 240 | 2007 |
| Synthesis of medium ring nitrogen heterocycles via a tandem copper-catalyzed C− N bond formation− ring-expansion process A Klapars, S Parris, KW Anderson, SL Buchwald Journal of the American Chemical Society 126 (11), 3529-3533, 2004 | 235 | 2004 |
| Palladium-catalyzed amination of aryl nonaflates KW Anderson, M Mendez-Perez, J Priego, SL Buchwald The Journal of Organic Chemistry 68 (25), 9563-9573, 2003 | 167 | 2003 |
| A Palladium‐Catalyzed Regiospecific Synthesis of N‐Aryl Benzimidazoles N Zheng, KW Anderson, X Huang, HN Nguyen, SL Buchwald Angewandte Chemie 119 (39), 7653-7656, 2007 | 164 | 2007 |
| Expedited palladium-catalyzed amination of aryl nonaflates through the use of microwave-irradiation and soluble organic amine bases RE Tundel, KW Anderson, SL Buchwald The Journal of Organic Chemistry 71 (1), 430-433, 2006 | 151 | 2006 |
| Pyrrole-2-carboxylic acid as a ligand for the Cu-catalyzed reactions of primary anilines with aryl halides RA Altman, KW Anderson, SL Buchwald The Journal of organic chemistry 73 (13), 5167-5169, 2008 | 97 | 2008 |
| Pyrido [2, 3-d] pyrimidines: discovery and preliminary SAR of a novel series of DYRK1B and DYRK1A inhibitors K Anderson, Y Chen, Z Chen, R Dominique, K Glenn, Y He, C Janson, ... Bioorganic & medicinal chemistry letters 23 (24), 6610-6615, 2013 | 60 | 2013 |
| Trifluoromethanesulfonic acid catalyzed Friedel–Crafts acylation of aromatics with β-lactams KW Anderson, JJ Tepe Tetrahedron 58 (42), 8475-8481, 2002 | 52 | 2002 |
| The first intermolecular Friedel− Crafts acylation with β-lactams KW Anderson, JJ Tepe Organic Letters 4 (3), 459-461, 2002 | 44 | 2002 |
| Palladium-catalyzed Heck alkynylation of benzyl chlorides CH Larsen, KW Anderson, RE Tundel, SL Buchwald Synlett 2006 (18), 2941-2946, 2006 | 36 | 2006 |
| Transition-metal-catalyzed carbon-nitrogen and carbon-carbon bond-forming reactions SL Buchwald, KW Anderson US Patent 7,560,596, 2009 | 14 | 2009 |
| Palladium-catalyzed decarboxylative benzylation of acetylides and enolates RRP Torregrosa, SN Mendis, A Davies, JA Tunge Synthesis 50 (16), 3205-3216, 2018 | 12 | 2018 |
| Pd/Indanone-Based Ligands: An Efficient Catalyst System for Ullmann-Type, Suzuki–Miyaura, and Mizoroki–Heck Cross-Coupling Reactions with Aryl Tosylates and Aryl Halides M Waheed, N Ahmed Synthesis 49 (18), 4372-4382, 2017 | 12 | 2017 |
| Transition-metal-catalyzed carbon-nitrogen and carbon-carbon bond-forming reactions SL Buchwald, KW Anderson US Patent 8,378,145, 2013 | 10 | 2013 |
| Preparation of Pyrazole-4-Carboxamide Derivatives as 11-β-Hydroxysteroid Dehydrogenase Form I (11-β-HSD1) Inhibitors KW Anderson, N Fotouhi, P Gillespie, RA Goodnow Jr, KR Guertin, ... World Patent WO2007107470A2, 2007 | 5 | 2007 |
Stephen L. BuchwaldProfessor of Chemistry, Massachusetts Institute of TechnologyVerified email at mit.edu
